Publikationer

Isaksson, Rebecka; Casselbrant, Anna; Elebring, Erik; Hallberg, Mathias et al.

Direct stimulation of angiotensin II type 2 receptor reduces nitric oxide production in lipopolysaccharide treated mouse macrophages

Ingår i European Journal of Pharmacology, 2020.

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Open access
Engen, Karin; Reddy Vanga, Sudarsana; Lundbäck, Thomas; Agalo, Faith et al.

Synthesis, Evaluation and Proposed Binding Pose of Substituted Spiro-Oxindole Dihydroquinazolinones as IRAP Inhibitors

Ingår i ChemistryOpen, s. 325-337, 2020.

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Open access
Barlow, Nicholas; Reddy Vanga, Sudarsana; Sävmarker, Jonas; Sandström, Anja et al.

Macrocyclic Peptidomimetics as Inhibitors of Insulin-Regulated Aminopeptidase (IRAP)

Ingår i RSC Medicinal chemistry, s. 234-244, 2020.

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Mpakali, Anastasia; Saridakis, Emmanuel; Giastas, Petros; Maben, Zachary et al.

Structural Basis of Inhibition of Insulin-Regulated Aminopeptidase by a Macrocyclic Peptidic Inhibitor

Ingår i ACS Medicinal Chemistry Letters, s. 1429-1434, 2020.

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Adeyemi, Ahmed; Odell, Luke R.; Larhed, Mats

Regio- and Stereoselective Synthesis of Allylic Spiroethers (Spirobenzofuranes) via an Intramolecular Mizoroki-Heck Reaction

Ingår i Journal of Organic Chemistry, s. 7648-7657, 2020.

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Open access
Lundmark, Fanny; Abouzayed, Ayman; Mitran, Bogdan; Rinne, Sara S. et al.

Heterodimeric Radiotracer Targeting PSMA and GRPR for Imaging of Prostate Cancer-Optimization of the Affinity towards PSMA by Linker Modification in Murine Model

Ingår i Pharmaceutics, 2020.

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Open access
Ye, Sofie; Hartmann, Rafael; Söderström, Marcus; Amin, Mohammad A. et al.

Turning Information Dissipation into Dissemination: Instagram as a Communication Enhancing Tool during the COVID-19 Pandemic and Beyond

Ingår i Journal of Chemical Education, s. 3217-3222, 2020.

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Hallberg, Mathias; Larhed, Mats

From Angiotensin IV to Small Peptidemimetics Inhibiting Insulin-Regulated Aminopeptidase

Ingår i Frontiers in Pharmacology, 2020.

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Open access
Isaksson, Rebecka; Lindman, Jens; Wannberg, Johan; Sallander, Jessica et al.

A Series of Analogues to the AT₂R Prototype Antagonist C38 Allow Fine Tuning of the Previously Reported Antagonist Binding Mode

Ingår i ChemistryOpen, s. 114-125, 2019.

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Open access
Schembri, Luke S; Eriksson, Jonas; Odell, Luke R.

Palladium(0)-Catalyzed Carbonylative Synthesis of N-Acylsulfonamides via Regioselective Acylation

Ingår i Journal of Organic Chemistry, s. 6970-6981, 2019.

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Eriksson, Jonas; Roy, Tamal; Sawadjoon, Supaporn; Bachmann, Kim et al.

Synthesis and preclinical evaluation of the CRTH2 antagonist [¹¹C]MK-7246 as a novel PET tracer and potential surrogate marker for pancreatic beta-cell mass

Ingår i Nuclear Medicine and Biology, s. 1-10, 2019.

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Open access
Abouzayed, Ayman; Yim, Cheng-Bin; Mitran, Bogdan; Rinne, Sara S. et al.

Synthesis and Preclinical Evaluation of Radio-Iodinated GRPR/PSMA Bispecific Heterodimers for the Theranostics Application in Prostate Cancer

Ingår i Pharmaceutics, 2019.

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Open access
Oroujeni, Maryam; Abouzayed, Ayman; Lundmark, Fanny; Mitran, Bogdan et al.

Evaluation of Tumor-Targeting Properties of an Antagonistic Bombesin Analogue RM26 Conjugated with a Non-Residualizing Radioiodine Label Comparison with a Radiometal-Labelled Counterpart

Ingår i Pharmaceutics, 2019.

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Open access
Söderström, Marcus; Zamaratski, Edouard; Odell, Luke R.

Thiomethylation, Nitro Reduction and Tandem Reduction/SMe Insertion of Nitrogen Heterocycles Using BF₃⦁SMe₂

Ingår i European Journal of Organic Chemistry, s. 5402-5408, 2019.

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Open access
Shariatgorji, Mohammadreza; Nilsson, Anna; Fridjonsdottir, Elva; Vallianatou, Theodosia et al.

Comprehensive mapping of neurotransmitter networks by MALDI-MS imaging

Ingår i Nature Methods, s. 1021-1028, 2019.

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Mitran, Bogdan; Rinne, Sara S.; Konijnenberg, Mark W.; Maina, Theodosia et al.

Trastuzumab cotreatment improves survival of mice with PC-3 prostate cancer xenografts treated with the GRPR antagonist 177Lu-DOTAGA-PEG2-RM26

Ingår i International Journal of Cancer, s. 3347-3358, 2019.

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Open access
Mitran, Bogdan; Thisgaard, Helge; Rinne, Sara S.; Dam, Johan Hygum et al.

Selection of an optimal macrocyclic chelator improves the imaging of prostate cancer using cobalt-labeled GRPR antagonist RM26

Ingår i Scientific Reports, 2019.

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Open access
Adeyemi, Ahmed; Wetzel, Alexander; Bergman, Joakim; Brånalt, Jonas et al.

Regio- and Stereoselective Synthesis of Spirooxindoles via Mizoroki-Heck Coupling of Aryl Iodides

Ingår i Synlett, s. 82-88, 2019.

DOI Till DiVA
Mitran, Bogdan; Varasteh, Zohreh; Abouzayed, Ayman; Rinne, Sara S. et al.

Bispecific GRPR-antagonistic anti-PSMA/GRPR heterodimer for PET and SPECT diagnostic imaging of prostate cancer

Ingår i Cancers, 2019.

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Open access
Åkerbladh, Linda; Odell, Luke R.; Larhed, Mats

Palladium-Catalyzed Molybdenum Hexacarbonyl-Mediated Gas-Free Carbonylative Reactions

Ingår i Synlett, s. 141-155, 2019.

DOI Till DiVA
Monazzam, Azita; Lau, Joey; Velikyan, Irina; Li, Su-Chen et al.

Increased Expression of GLP-1R in Proliferating Islets of Men1 Mice is Detectable by [Ga-68]Ga-DO3A-VS-Cys(40)- Exendin-4/PET

Ingår i Scientific Reports, 2018.

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Open access
Sawant, Rajiv T.; Stevens, Marc Y.; Odell, Luke R.

Microwave-Assisted aza-Friedel-Crafts Arylation of N-Acyliminium Ions: Expedient Access to 4 -Aryl 3,4-Dihydroquinazolinones

Ingår i ACS OMEGA, s. 14258 14258-14265 14265, 2018.

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Open access
Reddy Vanga, Sudarsana; Sävmarker, Jonas; Ng, Leelee; Larhed, Mats et al.

Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides

Ingår i ACS OMEGA, s. 4509 4509-4521 4521, 2018.

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Open access
Wannberg, Johan; Isaksson, Rebecka; Bremberg, Ulf; Backlund, Maria et al.

A convenient transesterification method for synthesis of AT2 receptor ligands with improved stability in human liver microsomes

Ingår i Bioorganic & Medicinal Chemistry Letters, s. 519-522, 2018.

DOI Till DiVA
Roy, Tamal; Brandt, Peter; Wetzel, Alexander; Bergman, Joakim et al.

Selective Synthesis of Spirooxindoles by an Intramolecular Heck-Mizoroki Reaction

Ingår i Organic Letters, s. 2738-2741, 2017.

DOI Till DiVA
Roslin, Sara; Odell, Luke R.

Visible-Light Photocatalysis as an Enabling Tool for the Functionalization of Unactivated C(sp(3))-Substrates

Ingår i European Journal of Organic Chemistry, s. 1993-2007, 2017.

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Velikyan, Irina; Rosenström, Ulrika; Eriksson, Olof

Fully automated GMP production of [Ga-68]Ga-DO3A-VS-Cys(40)-Exendin-4 for clinical use

Ingår i American Journal of Nuclear Medicine and Molecular Imaging, s. 111-125, 2017.

Uppladdad fulltext Till DiVA

Open access
Chow, Shiao Y.; Odell, Luke R.

Synthesis of N-Sulfonyl Amidines and Acyl Sulfonyl Ureas from Sulfonyl Azides, Carbon Monoxide, and Amides

Ingår i Journal of Organic Chemistry, s. 2515-2522, 2017.

DOI Till DiVA
Sawant, Rajiv T.; Stevens, Marc Y.; Odell, Luke R.

Acetic acid-promoted cascade N-acyliminium ion/aza-Prins cyclization: stereoselective synthesis of functionalized fused tricyclic piperidines

Ingår i Chemical Communications, s. 2110-2113, 2017.

DOI Till DiVA
Wetzel, Alexander; Bergman, Joakim; Brandt, Peter; Larhed, Mats et al.

Regio- and Stereoselective Synthesis of Functionalized Cyclopentene Derivatives via Mizoroki-Heck Reactions.

Ingår i Organic Letters, s. 1602-1605, 2017.

DOI Till DiVA

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Publikationer

Direct stimulation of angiotensin II type 2 receptor reduces nitric oxide production in lipopolysaccharide treated mouse macrophages

Synthesis, Evaluation and Proposed Binding Pose of Substituted Spiro-Oxindole Dihydroquinazolinones as IRAP Inhibitors

Macrocyclic Peptidomimetics as Inhibitors of Insulin-Regulated Aminopeptidase (IRAP)

Structural Basis of Inhibition of Insulin-Regulated Aminopeptidase by a Macrocyclic Peptidic Inhibitor

Regio- and Stereoselective Synthesis of Allylic Spiroethers (Spirobenzofuranes) via an Intramolecular Mizoroki-Heck Reaction

Heterodimeric Radiotracer Targeting PSMA and GRPR for Imaging of Prostate Cancer-Optimization of the Affinity towards PSMA by Linker Modification in Murine Model

Turning Information Dissipation into Dissemination: Instagram as a Communication Enhancing Tool during the COVID-19 Pandemic and Beyond

From Angiotensin IV to Small Peptidemimetics Inhibiting Insulin-Regulated Aminopeptidase

A Series of Analogues to the AT2R Prototype Antagonist C38 Allow Fine Tuning of the Previously Reported Antagonist Binding Mode

Palladium(0)-Catalyzed Carbonylative Synthesis of N-Acylsulfonamides via Regioselective Acylation

Synthesis and preclinical evaluation of the CRTH2 antagonist [11C]MK-7246 as a novel PET tracer and potential surrogate marker for pancreatic beta-cell mass

Synthesis and Preclinical Evaluation of Radio-Iodinated GRPR/PSMA Bispecific Heterodimers for the Theranostics Application in Prostate Cancer

Evaluation of Tumor-Targeting Properties of an Antagonistic Bombesin Analogue RM26 Conjugated with a Non-Residualizing Radioiodine Label Comparison with a Radiometal-Labelled Counterpart

Thiomethylation, Nitro Reduction and Tandem Reduction/SMe Insertion of Nitrogen Heterocycles Using BF3⦁SMe2

Comprehensive mapping of neurotransmitter networks by MALDI-MS imaging

Trastuzumab cotreatment improves survival of mice with PC-3 prostate cancer xenografts treated with the GRPR antagonist 177Lu-DOTAGA-PEG2-RM26

Selection of an optimal macrocyclic chelator improves the imaging of prostate cancer using cobalt-labeled GRPR antagonist RM26

Regio- and Stereoselective Synthesis of Spirooxindoles via Mizoroki-Heck Coupling of Aryl Iodides

Bispecific GRPR-antagonistic anti-PSMA/GRPR heterodimer for PET and SPECT diagnostic imaging of prostate cancer

Palladium-Catalyzed Molybdenum Hexacarbonyl-Mediated Gas-Free Carbonylative Reactions

Increased Expression of GLP-1R in Proliferating Islets of Men1 Mice is Detectable by [Ga-68]Ga-DO3A-VS-Cys(40)- Exendin-4/PET

Microwave-Assisted aza-Friedel-Crafts Arylation of N-Acyliminium Ions: Expedient Access to 4 -Aryl 3,4-Dihydroquinazolinones

Structural Basis of Inhibition of Human Insulin-Regulated Aminopeptidase (IRAP) by Aryl Sulfonamides

A convenient transesterification method for synthesis of AT2 receptor ligands with improved stability in human liver microsomes

Selective Synthesis of Spirooxindoles by an Intramolecular Heck-Mizoroki Reaction

Visible-Light Photocatalysis as an Enabling Tool for the Functionalization of Unactivated C(sp(3))-Substrates

Fully automated GMP production of [Ga-68]Ga-DO3A-VS-Cys(40)-Exendin-4 for clinical use

Synthesis of N-Sulfonyl Amidines and Acyl Sulfonyl Ureas from Sulfonyl Azides, Carbon Monoxide, and Amides

Acetic acid-promoted cascade N-acyliminium ion/aza-Prins cyclization: stereoselective synthesis of functionalized fused tricyclic piperidines

Regio- and Stereoselective Synthesis of Functionalized Cyclopentene Derivatives via Mizoroki-Heck Reactions.

A Series of Analogues to the AT₂R Prototype Antagonist C38 Allow Fine Tuning of the Previously Reported Antagonist Binding Mode

Synthesis and preclinical evaluation of the CRTH2 antagonist [¹¹C]MK-7246 as a novel PET tracer and potential surrogate marker for pancreatic beta-cell mass

Thiomethylation, Nitro Reduction and Tandem Reduction/SMe Insertion of Nitrogen Heterocycles Using BF₃⦁SMe₂