Publikationer
-
Green multifunctional palladium nanoparticles from polysaccharide cordia myxa (CMY) gum: Synthesis, characterization, and antibacterial activity
Ingår i Colloids and Surfaces A, 2023.
-
Söderström, Marcus
C1 Building Blocks: New Approaches for Thiomethylations and Esterification
A1:111a, BMC, Husargatan 3, Uppsala 2023-12-20 kl 13:15
-
Thioacetalation and Multi-Component Thiomethylative Friedel-Crafts Arylation Using BF3SMe2
Ingår i ACS Omega, s. 4320-4330, 2023.
DOI för Thioacetalation and Multi-Component Thiomethylative Friedel-Crafts Arylation Using BF3SMe2 Ladda ner fulltext (pdf) av Thioacetalation and Multi-Component Thiomethylative Friedel-Crafts Arylation Using BF3SMe2
-
Bifunctional and regenerable molecular electrode for water electrolysis at neutral pH
Ingår i Journal of Materials Chemistry A, s. 13331-13340, 2023.
DOI för Bifunctional and regenerable molecular electrode for water electrolysis at neutral pH Ladda ner fulltext (pdf) av Bifunctional and regenerable molecular electrode for water electrolysis at neutral pH
-
A Base-Free, Low Temperature Click and Release Reaction for the In Situ Generation of Diazomethane
Ingår i Advanced Synthesis and Catalysis, s. 1839-1845, 2023.
DOI för A Base-Free, Low Temperature Click and Release Reaction for the In Situ Generation of Diazomethane Ladda ner fulltext (pdf) av A Base-Free, Low Temperature Click and Release Reaction for the In Situ Generation of Diazomethane
-
Antimicrobial Peptides Incorporating Halogenated Marine-Derived Amino Acid Substituents
Ingår i ACS Medicinal Chemistry Letters, s. 802-809, 2023.
DOI för Antimicrobial Peptides Incorporating Halogenated Marine-Derived Amino Acid Substituents
-
Hybrid Machine Learning Approach to Predict the Site Selectivity of Iridium-Catalyzed Arene Borylation
Ingår i Journal of the American Chemical Society, s. 17367-17376, 2023.
-
Characterization of a Newly Available Coastal Marine Dissolved Organic Matter Reference Material (TRM-0522)
Ingår i Analytical Chemistry, s. 6559-6567, 2023.
DOI för Characterization of a Newly Available Coastal Marine Dissolved Organic Matter Reference Material (TRM-0522) Ladda ner fulltext (pdf) av Characterization of a Newly Available Coastal Marine Dissolved Organic Matter Reference Material (TRM-0522)
-
Influence of extracellular matrix composition on tumour cell behaviour in a biomimetic in vitro model for hepatocellular carcinoma
Ingår i Scientific Reports, 2023.
DOI för Influence of extracellular matrix composition on tumour cell behaviour in a biomimetic in vitro model for hepatocellular carcinoma Ladda ner fulltext (pdf) av Influence of extracellular matrix composition on tumour cell behaviour in a biomimetic in vitro model for hepatocellular carcinoma
-
Physiologically based biopharmaceutics modeling of regional and colon absorption in humans
Ingår i European journal of pharmaceutics and biopharmaceutics, s. 144-159, 2023.
DOI för Physiologically based biopharmaceutics modeling of regional and colon absorption in humans
-
On-Tissue Chemical Derivatization for Comprehensive Mapping of Brain Carboxyl and Aldehyde Metabolites by MALDI-MS Imaging
Ingår i Journal of the American Society for Mass Spectrometry, s. 836-846, 2023.
DOI för On-Tissue Chemical Derivatization for Comprehensive Mapping of Brain Carboxyl and Aldehyde Metabolites by MALDI-MS Imaging Ladda ner fulltext (pdf) av On-Tissue Chemical Derivatization for Comprehensive Mapping of Brain Carboxyl and Aldehyde Metabolites by MALDI-MS Imaging
-
Novel food drug interaction mechanism involving acyclovir, chitosan and endogenous mucus
Ingår i Drug Metabolism and Pharmacokinetics, 2023.
DOI för Novel food drug interaction mechanism involving acyclovir, chitosan and endogenous mucus
-
SPICY: a method for single scan rotating frame relaxometry
Ingår i Physical Chemistry, Chemical Physics - PCCP, s. 13164-13169, 2023.
DOI för SPICY: a method for single scan rotating frame relaxometry Ladda ner fulltext (pdf) av SPICY: a method for single scan rotating frame relaxometry
-
[18F]MK-7246 for Positron Emission Tomography Imaging of the Beta-Cell Surface Marker GPR44
Ingår i Pharmaceutics, 2023.
DOI för [18F]MK-7246 for Positron Emission Tomography Imaging of the Beta-Cell Surface Marker GPR44 Ladda ner fulltext (pdf) av [18F]MK-7246 for Positron Emission Tomography Imaging of the Beta-Cell Surface Marker GPR44
-
Electrochemical Palladium-Catalyzed Oxidative Carbonylation-Cyclization of Enallenols
Ingår i Angewandte Chemie International Edition, 2022.
DOI för Electrochemical Palladium-Catalyzed Oxidative Carbonylation-Cyclization of Enallenols Ladda ner fulltext (pdf) av Electrochemical Palladium-Catalyzed Oxidative Carbonylation-Cyclization of Enallenols
-
Novel Allosteric Mechanism of Dual p53/MDM2 and p53/MDM4 Inhibition by a Small Molecule
Ingår i Frontiers in Molecular Biosciences, 2022.
DOI för Novel Allosteric Mechanism of Dual p53/MDM2 and p53/MDM4 Inhibition by a Small Molecule Ladda ner fulltext (pdf) av Novel Allosteric Mechanism of Dual p53/MDM2 and p53/MDM4 Inhibition by a Small Molecule
-
Bacterial type I signal peptidase inhibitors-Optimized hits from nature
Ingår i European Journal of Medicinal Chemistry, 2022.
DOI för Bacterial type I signal peptidase inhibitors-Optimized hits from nature
-
2-Alkyl substituted benzimidazoles as a new class of selective AT2 receptor ligands
Ingår i Bioorganic & Medicinal Chemistry, 2022.
DOI för 2-Alkyl substituted benzimidazoles as a new class of selective AT2 receptor ligands Ladda ner fulltext (pdf) av 2-Alkyl substituted benzimidazoles as a new class of selective AT2 receptor ligands
-
Protective Effects of Melatonin and Misoprostol against Experimentally Induced Increases in Intestinal Permeability in Rats
Ingår i International Journal of Molecular Sciences, 2022.
DOI för Protective Effects of Melatonin and Misoprostol against Experimentally Induced Increases in Intestinal Permeability in Rats Ladda ner fulltext (pdf) av Protective Effects of Melatonin and Misoprostol against Experimentally Induced Increases in Intestinal Permeability in Rats
-
Ultralarge Virtual Screening Identifies SARS-CoV-2 Main Protease Inhibitors with Broad-Spectrum Activity against Coronaviruses
Ingår i Journal of the American Chemical Society, s. 2905-2920, 2022.
DOI för Ultralarge Virtual Screening Identifies SARS-CoV-2 Main Protease Inhibitors with Broad-Spectrum Activity against Coronaviruses Ladda ner fulltext (pdf) av Ultralarge Virtual Screening Identifies SARS-CoV-2 Main Protease Inhibitors with Broad-Spectrum Activity against Coronaviruses
-
Dipolar Relaxation of Water Protons in the Vicinity of a Collagen-like Peptide
Ingår i Journal of Physical Chemistry B, s. 2538-2551, 2022.
DOI för Dipolar Relaxation of Water Protons in the Vicinity of a Collagen-like Peptide Ladda ner fulltext (pdf) av Dipolar Relaxation of Water Protons in the Vicinity of a Collagen-like Peptide
-
Spatial Distribution and Stability of Cholinesterase Inhibitory Protoberberine Alkaloids from Papaver setiferum
Ingår i Journal of Natural Products, s. 215-224, 2022.
DOI för Spatial Distribution and Stability of Cholinesterase Inhibitory Protoberberine Alkaloids from Papaver setiferum Ladda ner fulltext (pdf) av Spatial Distribution and Stability of Cholinesterase Inhibitory Protoberberine Alkaloids from Papaver setiferum
-
Chemotherapeutics Combined with Luminal Irritants: Effects on Small-Intestinal Mannitol Permeability and Villus Length in Rats
Ingår i International Journal of Molecular Sciences, 2022.
DOI för Chemotherapeutics Combined with Luminal Irritants: Effects on Small-Intestinal Mannitol Permeability and Villus Length in Rats Ladda ner fulltext (pdf) av Chemotherapeutics Combined with Luminal Irritants: Effects on Small-Intestinal Mannitol Permeability and Villus Length in Rats
-
Synthesis and in vitro biological evaluation of quinolinyl pyrimidines targeting type II NADH-dehydrogenase (NDH-2)
Ingår i ACS Infectious Diseases, s. 482-498, 2022.
DOI för Synthesis and in vitro biological evaluation of quinolinyl pyrimidines targeting type II NADH-dehydrogenase (NDH-2) Ladda ner fulltext (pdf) av Synthesis and in vitro biological evaluation of quinolinyl pyrimidines targeting type II NADH-dehydrogenase (NDH-2)
-
Towards the sustainable discovery and development of new antibiotics
Ingår i Nature Reviews Chemistry, s. 726-749, 2021.
DOI för Towards the sustainable discovery and development of new antibiotics
-
A Genetically Encoded Picolyl Azide for Improved Live Cell Copper Click Labeling
Ingår i Frontiers in Chemistry, 2021.
DOI för A Genetically Encoded Picolyl Azide for Improved Live Cell Copper Click Labeling Ladda ner fulltext (pdf) av A Genetically Encoded Picolyl Azide for Improved Live Cell Copper Click Labeling
-
Influence of Detergent and Lipid Composition on Reconstituted Membrane Proteins for Structural Studies
Ingår i ACS Omega, s. 24377-24381, 2021.
DOI för Influence of Detergent and Lipid Composition on Reconstituted Membrane Proteins for Structural Studies Ladda ner fulltext (pdf) av Influence of Detergent and Lipid Composition on Reconstituted Membrane Proteins for Structural Studies
-
The Impact of Ligand Carboxylates on Electrocatalyzed Water Oxidation
Ingår i Accounts of Chemical Research, s. 3326-3337, 2021.
DOI för The Impact of Ligand Carboxylates on Electrocatalyzed Water Oxidation Ladda ner fulltext (pdf) av The Impact of Ligand Carboxylates on Electrocatalyzed Water Oxidation
-
Organic reactivity from mechanism to machine learning
Ingår i Nature Reviews Chemistry, s. 240-255, 2021.
DOI för Organic reactivity from mechanism to machine learning
-
A Study of an 8-Aminoquinoline-Directed C(sp(2))-H Arylation Reaction on the Route to Chiral Cyclobutane Keto Acids from Myrtenal
Ingår i Journal of Organic Chemistry, s. 8527-8537, 2021.
DOI för A Study of an 8-Aminoquinoline-Directed C(sp(2))-H Arylation Reaction on the Route to Chiral Cyclobutane Keto Acids from Myrtenal Ladda ner fulltext (pdf) av A Study of an 8-Aminoquinoline-Directed C(sp(2))-H Arylation Reaction on the Route to Chiral Cyclobutane Keto Acids from Myrtenal
-
Antibacterial sulfonimidamide-based oligopeptides as type I signal peptidase inhibitors: Synthesis and biological evaluation
Ingår i European Journal of Medicinal Chemistry, 2021.
DOI för Antibacterial sulfonimidamide-based oligopeptides as type I signal peptidase inhibitors: Synthesis and biological evaluation Ladda ner fulltext (pdf) av Antibacterial sulfonimidamide-based oligopeptides as type I signal peptidase inhibitors: Synthesis and biological evaluation
-
ENABLE: an engine for European antibacterial drug discovery and development
Ingår i Nature reviews. Drug discovery, s. 407-408, 2021.
DOI för ENABLE: an engine for European antibacterial drug discovery and development
-
Computational studies of molecular pre-organization through macrocyclization: Conformational distribution analysis of closely related non-macrocyclic and macrocyclic analogs
Ingår i Bioorganic & Medicinal Chemistry, 2021.
DOI för Computational studies of molecular pre-organization through macrocyclization: Conformational distribution analysis of closely related non-macrocyclic and macrocyclic analogs Ladda ner fulltext (pdf) av Computational studies of molecular pre-organization through macrocyclization: Conformational distribution analysis of closely related non-macrocyclic and macrocyclic analogs
-
Investigation of the Deactivation and Reactivation Mechanism of a Heterogeneous Palladium(II) Catalyst in the Cycloisomerization of Acetylenic Acids by In Situ XAS
Ingår i ACS Catalysis, s. 2999-3008, 2021.
DOI för Investigation of the Deactivation and Reactivation Mechanism of a Heterogeneous Palladium(II) Catalyst in the Cycloisomerization of Acetylenic Acids by In Situ XAS Ladda ner fulltext (pdf) av Investigation of the Deactivation and Reactivation Mechanism of a Heterogeneous Palladium(II) Catalyst in the Cycloisomerization of Acetylenic Acids by In Situ XAS
-
Enantioselective Synthesis of Atropisomeric Biaryls using Biaryl 2,5-Diphenylphospholanes as Ligands for Palladium-Catalysed Suzuki-Miyaura Reactions
Ingår i Advanced Synthesis and Catalysis, s. 259-267, 2021.
-
The amino-terminal heptapeptide of the algesic substance P provides analgesic effect in relieving chronic neuropathic pain
Ingår i European Journal of Pharmacology, 2021.
-
Characterization of More Selective Central Nervous System Nrf2-Activating Novel Vinyl Sulfoximine Compounds Compared to Dimethyl Fumarate
Ingår i NEUROTHERAPEUTICS, s. 1142-1152, 2020.
DOI för Characterization of More Selective Central Nervous System Nrf2-Activating Novel Vinyl Sulfoximine Compounds Compared to Dimethyl Fumarate Ladda ner fulltext (pdf) av Characterization of More Selective Central Nervous System Nrf2-Activating Novel Vinyl Sulfoximine Compounds Compared to Dimethyl Fumarate
-
Nanocatalysis Meets Biology
Ingår i Nanoparticles in catalysis, s. 243-278, 2020.
-
Phidianidine A and Synthetic Analogues as Naturally Inspired Marine Antifoulants
Ingår i Journal of Natural Products, s. 3413-3423, 2020.
DOI för Phidianidine A and Synthetic Analogues as Naturally Inspired Marine Antifoulants
-
Identification of a C2-symmetric diol based human immunodeficiency virus protease inhibitor targeting Zika virus NS2B-NS3 protease
Ingår i Journal of Biomolecular Structure and Dynamics, s. 5526-5536, 2020.
DOI för Identification of a C2-symmetric diol based human immunodeficiency virus protease inhibitor targeting Zika virus NS2B-NS3 protease Ladda ner fulltext (pdf) av Identification of a C2-symmetric diol based human immunodeficiency virus protease inhibitor targeting Zika virus NS2B-NS3 protease
-
Intestinal absorption of BCS class II drugs administered as nanoparticles: A review based on in vivo data from intestinal perfusion models
Ingår i ADMET & DMPK, s. 375-390, 2020.
DOI för Intestinal absorption of BCS class II drugs administered as nanoparticles: A review based on in vivo data from intestinal perfusion models Ladda ner fulltext (pdf) av Intestinal absorption of BCS class II drugs administered as nanoparticles: A review based on in vivo data from intestinal perfusion models
-
Turning Information Dissipation into Dissemination: Instagram as a Communication Enhancing Tool during the COVID-19 Pandemic and Beyond
Ingår i Journal of Chemical Education, s. 3217-3222, 2020.
-
Sulfadiazine Masquerading as a Natural Product from Scilla madeirensis (Scilloideae)
Ingår i Journal of Natural Products, s. 1305-1308, 2020.
DOI för Sulfadiazine Masquerading as a Natural Product from Scilla madeirensis (Scilloideae) Ladda ner fulltext (pdf) av Sulfadiazine Masquerading as a Natural Product from Scilla madeirensis (Scilloideae)
-
The global preclinical antibacterial pipeline
Ingår i Nature Reviews Microbiology, s. 275-285, 2020.
-
Solid Phase Synthesis of Sulfonimidamide Pseudopeptides and Library Generation
Ingår i European Journal of Organic Chemistry, s. 3796-3807, 2020.
DOI för Solid Phase Synthesis of Sulfonimidamide Pseudopeptides and Library Generation Ladda ner fulltext (pdf) av Solid Phase Synthesis of Sulfonimidamide Pseudopeptides and Library Generation
-
Synthesis, Evaluation and Proposed Binding Pose of Substituted Spiro-Oxindole Dihydroquinazolinones as IRAP Inhibitors
Ingår i ChemistryOpen, s. 325-337, 2020.
DOI för Synthesis, Evaluation and Proposed Binding Pose of Substituted Spiro-Oxindole Dihydroquinazolinones as IRAP Inhibitors Ladda ner fulltext (pdf) av Synthesis, Evaluation and Proposed Binding Pose of Substituted Spiro-Oxindole Dihydroquinazolinones as IRAP Inhibitors
-
Macrocyclic Peptidomimetics as Inhibitors of Insulin-Regulated Aminopeptidase (IRAP)
Ingår i RSC Medicinal chemistry, s. 234-244, 2020.
DOI för Macrocyclic Peptidomimetics as Inhibitors of Insulin-Regulated Aminopeptidase (IRAP)
-
Conformational Analysis of Macrocycles: Comparing General and Specialized Methods
Ingår i Journal of Computer-Aided Molecular Design, s. 231-252, 2020.
DOI för Conformational Analysis of Macrocycles: Comparing General and Specialized Methods Ladda ner fulltext (pdf) av Conformational Analysis of Macrocycles: Comparing General and Specialized Methods
-
Relative Strength of Common Directing Groups in Palladium-Catalyzed Aromatic C-H Activation
Ingår i iScience, s. 373-+, 2019.
DOI för Relative Strength of Common Directing Groups in Palladium-Catalyzed Aromatic C-H Activation Ladda ner fulltext (pdf) av Relative Strength of Common Directing Groups in Palladium-Catalyzed Aromatic C-H Activation
-
Cellular uptake of self-assembled phytantriol-based hexosomes is independent of major endocytic machineries
Ingår i Journal of Colloid and Interface Science, s. 820-833, 2019.
-
Thiomethylation, Nitro Reduction and Tandem Reduction/SMe Insertion of Nitrogen Heterocycles Using BF3⦁SMe2
Ingår i European Journal of Organic Chemistry, s. 5402-5408, 2019.
DOI för Thiomethylation, Nitro Reduction and Tandem Reduction/SMe Insertion of Nitrogen Heterocycles Using BF3⦁SMe2 Ladda ner fulltext (pdf) av Thiomethylation, Nitro Reduction and Tandem Reduction/SMe Insertion of Nitrogen Heterocycles Using BF3⦁SMe2
-
Synthesis and preclinical evaluation of the CRTH2 antagonist [11C]MK-7246 as a novel PET tracer and potential surrogate marker for pancreatic beta-cell mass
Ingår i Nuclear Medicine and Biology, s. 1-10, 2019.
DOI för Synthesis and preclinical evaluation of the CRTH2 antagonist [11C]MK-7246 as a novel PET tracer and potential surrogate marker for pancreatic beta-cell mass Ladda ner fulltext (pdf) av Synthesis and preclinical evaluation of the CRTH2 antagonist [11C]MK-7246 as a novel PET tracer and potential surrogate marker for pancreatic beta-cell mass
-
Synthesis of Sulfonimidamide-Based Amino Acid Building Blocks with Orthogonal Protecting Groups
Ingår i European Journal of Organic Chemistry, s. 1045-1057, 2019.
-
From the Anti-Nociceptive Substance P Metabolite Substance P (1-7) to Small Peptidomimetics
Ingår i Current protein and peptide science, s. 1038-1048, 2018.
DOI för From the Anti-Nociceptive Substance P Metabolite Substance P (1-7) to Small Peptidomimetics
-
Sulfonyl Fluorides (SFs): More Than Click Reagents?
Ingår i European Journal of Organic Chemistry, s. 3648-3666, 2018.
-
Boronic ester-linked macrocyclic lipopeptides as serine protease inhibitors targeting Escherichia coli type I signal peptidase
Ingår i European Journal of Medicinal Chemistry, s. 1346-1360, 2018.
-
An imidazole based H-Phe-Phe-NH2 peptidomimetic with anti-allodynic effect in spared nerve injury mice
Ingår i Bioorganic & Medicinal Chemistry Letters, s. 2446-2450, 2018.
-
Pan-NS3 protease inhibitors of hepatitis C virus based on an R3-elongated pyrazinone scaffold
Ingår i European Journal of Medicinal Chemistry, s. 453-464, 2018.
-
Impact of N-methylation of the substance P 1-7 amide on anti-allodynic effect in mice after peripheral administration
Ingår i European Journal of Pharmaceutical Sciences, s. 533-540, 2017.
-
Importance of N-and C-terminal residues of substance P 1-7 for alleviating allodynia in mice after peripheral administration
Ingår i European Journal of Pharmaceutical Sciences, s. 345-351, 2017.
-
Palladium-Catalyzed Aminocarbonylation in Solid-Phase Peptide Synthesis: A Method for Capping, Cyclization, and Isotope Labeling
Ingår i Organic Letters, s. 2873-2876, 2017.
-
Predicting the Rate of Skin Penetration Using an Aggregated Conformal Prediction Framework
Ingår i Molecular Pharmaceutics, s. 1571-1576, 2017.
DOI för Predicting the Rate of Skin Penetration Using an Aggregated Conformal Prediction Framework
-
Docking of Macrocycles: Comparing Rigid and Flexible Docking in Glide
Ingår i Journal of Chemical Information and Modeling, s. 190-202, 2017.
DOI för Docking of Macrocycles: Comparing Rigid and Flexible Docking in Glide
-
Design, synthesis and in vitro biological evaluation of oligopeptides targeting E. coli type I signal peptidase (LepB)
Ingår i Bioorganic & Medicinal Chemistry, s. 897-911, 2017.
DOI för Design, synthesis and in vitro biological evaluation of oligopeptides targeting E. coli type I signal peptidase (LepB) Ladda ner fulltext (pdf) av Design, synthesis and in vitro biological evaluation of oligopeptides targeting E. coli type I signal peptidase (LepB)
-
The Innovative Medicines Initiative's New Drugs for Bad Bugs programme: European public-private partnerships for the development of new strategies to tackle antibiotic resistance
Ingår i Journal of Antimicrobial Chemotherapy, s. 290-295, 2016.
-
Structural determinants of subtype selectivity and functional activity of angiotensin II receptors
Ingår i Bioorganic & Medicinal Chemistry Letters, s. 1355-1359, 2016.
-
Discovery of pyrazinone based compounds that potently inhibit the drug resistant enzyme variant R155K of the hepatitis C virus NS3 protease
Ingår i Bioorganic & Medicinal Chemistry, s. 2603-2620, 2016.
-
Palladium-Catalyzed Carbonylation of Aryl Iodides with Sulfinamides
Ingår i European Journal of Organic Chemistry, s. 7069-7074, 2015.
DOI för Palladium-Catalyzed Carbonylation of Aryl Iodides with Sulfinamides
-
Virtual Screening for Transition State Analogue Inhibitors of IRAP Based on Quantum Mechanically Derived Reaction Coordinates
Ingår i Journal of Chemical Information and Modeling, s. 1984-1993, 2015.
-
Optimization and Evaluation of 5-Styryl-Oxathiazol-2-one Mycobacterium tuberculosis Proteasome Inhibitors as Potential Antitubercular Agents
Ingår i ChemistryOpen, s. 342-362, 2015.
DOI för Optimization and Evaluation of 5-Styryl-Oxathiazol-2-one Mycobacterium tuberculosis Proteasome Inhibitors as Potential Antitubercular Agents Ladda ner fulltext (pdf) av Optimization and Evaluation of 5-Styryl-Oxathiazol-2-one Mycobacterium tuberculosis Proteasome Inhibitors as Potential Antitubercular Agents
-
Toward a Benchmarking Data Set Able to Evaluate Ligand- and Structure-based Virtual Screening Using Public HTS Data
Ingår i Journal of Chemical Information and Modeling, s. 343-353, 2015.
-
Small constrained SP1-7 analogues bind to a unique site and promote anti-allodynic effects following systemic injection in mice
Ingår i Neuroscience, s. 112-119, 2015.
-
Efficient and Selective Palladium-Catalysed C-3 Urea Couplings to 3,5-Dichloro-2(1H)-pyrazinones
Ingår i European Journal of Organic Chemistry, s. 978-986, 2015.
-
Synthesis of Vinyl- and Aryl–Acyl Sulfonimidamides Through Pd-Catalyzed Carbonylation Using Mo(CO)6 as ex situ CO Source
Ingår i European Journal of Organic Chemistry, s. 213-219, 2015.
-
Phototriggerable peptidomimetics for the inhibition of Mycobacterium turberculosis ribonucleotide reductase by targeting protein-protein binding
Ingår i Organic and biomolecular chemistry, s. 2612-2621, 2015.
-
Interconversion of Functional Activity by Minor Structural Alterations in Nonpeptide AT2 Receptor Ligands
Ingår i ACS Medicinal Chemistry Letters, s. 178-182, 2015.
-
Palladium(II) catalyzed desulfitative coupling reactions of sodium aryl sulfinates and nitriles: Scope, limitations, and mechanistic studies
Ingår i Abstracts of Papers of the American Chemical Society, 2014.
-
Inhibition of Insulin-Regulated Aminopeptidase (IRAP) by Arylsulfonamides
Ingår i ChemistryOpen, s. 256-263, 2014.
DOI för Inhibition of Insulin-Regulated Aminopeptidase (IRAP) by Arylsulfonamides
-
Palladium(II)-Catalyzed Desulfitative Synthesis of Aryl Ketones from Sodium Arylsulfinates and Nitriles: Scope, Limitations, and Mechanistic Studies
Ingår i Journal of Organic Chemistry, s. 12018-12032, 2014.
-
Exploration and pharmacokinetic profiling of phenylalanine based carbamates as novel substance p 1-7 analogues
Ingår i ACS Medicinal Chemistry Letters, s. 1272-1277, 2014.
-
Vinylated linear P2 pyrimidinyloxyphenylglycine based inhibitors of the HCV NS3/4A protease and corresponding macrocycles
Ingår i Bioorganic & Medicinal Chemistry, s. 6595-6615, 2014.
-
Saralasin and Sarile Are AT2 Receptor Agonists
Ingår i ACS Medicinal Chemistry Letters, s. 1129-1132, 2014.
-
N-terminal truncations of substance P1-7 amide affect its action on spinal cord injury-induced mechanical allodynia in rats
Ingår i European Journal of Pharmacology, s. 319-325, 2014.
-
Discovery and preclinical development of new antibiotics
Ingår i Upsala Journal of Medical Sciences, s. 162-169, 2014.
DOI för Discovery and preclinical development of new antibiotics
-
Novel Peptidomimetic Hepatitis C Virus NS3/4A Protease Inhibitors Spanning the P2–P1′ Region
Ingår i ACS Medicinal Chemistry Letters, s. 249-254, 2014.
DOI för Novel Peptidomimetic Hepatitis C Virus NS3/4A Protease Inhibitors Spanning the P2–P1′ Region
-
Synthesis and evaluation of isoleucine derived angiotensin II AT(2) receptor ligands
Ingår i Bioorganic & Medicinal Chemistry Letters, s. 476-479, 2014.
DOI för Synthesis and evaluation of isoleucine derived angiotensin II AT(2) receptor ligands
-
Achiral Pyrazinone-Based Inhibitors of the Hepatitis C Virus NS3 Protease and Drug-Resistant Variants with Elongated Substituents Directed Toward the S2 Pocket
Ingår i Journal of Medicinal Chemistry, s. 1790-1801, 2014.
-
Aminocarbonylation of 4-Iodo-1H-imidazoles with an Amino Acid Amide Nucleophile: Synthesis of Constrained H-Phe-Phe-NH2 Analogues
Ingår i Journal of Organic Chemistry, s. 12251-12256, 2013.
-
Decarboxylative Palladium(II)-Catalyzed Synthesis of Aryl Amidines from Aryl Carboxylic Acids: Development and Mechanistic Investigation
Ingår i Chemistry - A European Journal, s. 13803-13810, 2013.
-
One-Pot, Two-Step, Microwave-Assisted Palladium-Catalyzed Conversion of Aryl Alcohols to Aryl Fluorides via Aryl Nonaflates
Ingår i Journal of Organic Chemistry, s. 4184-4189, 2013.
-
DXR Inhibition by Potent Mono- and Disubstituted Fosmidomycin Analogues
Ingår i Journal of Medicinal Chemistry, s. 6190-6199, 2013.
DOI för DXR Inhibition by Potent Mono- and Disubstituted Fosmidomycin Analogues Ladda ner fulltext (pdf) av DXR Inhibition by Potent Mono- and Disubstituted Fosmidomycin Analogues
-
Theoretical and Experimental Investigation of Palladium(II)-Catalyzed Decarboxylative Addition of Arenecarboxylic Acid to Nitrile
Ingår i Organometallics, s. 490-497, 2013.
-
Angiotensin II type 2 receptor promotes adipocyte differentiation and restores adipocyte size in high-fat/high-fructose diet-induced insulin resistance in rats
Ingår i American Journal of Physiology. Endocrinology and Metabolism, s. E197-E210, 2013.
-
Constrained H-Phe-Phe-NH2 Analogues With High Affinity to the Substance P 1-7 Binding Site and With Improved Metabolic Stability and Cell Permeability
Ingår i Journal of Medicinal Chemistry, s. 4953-4965, 2013.
-
Novel pseudopeptides incorporating a benzodiazepine-based turn mimetic – targeting Mycobacterium tuberculosis ribonucleotide reductase
Ingår i Bioorganic & Medicinal Chemistry, s. 1992-2000, 2013.
-
AT2 Receptor Agonists: Exploiting the Beneficial Arm of Ang II Signaling
Ingår i current hypertension reviews, s. 47-59, 2012.
DOI för AT2 Receptor Agonists: Exploiting the Beneficial Arm of Ang II Signaling
-
Comparative functional properties of two structurally similar selective nonpeptide drug-like ligands for the angiotensin II type-2 (AT2) receptor. Effects on neurite outgrowth in NG108-15 cells
Ingår i European Journal of Pharmacology - Molecular Pharmacology Section, s. 160-171, 2012.
-
Use of Peptides as Drug Leads: A Case Story on the Development of Dipeptides Corresponding to the Heptapeptide Substance P(1-7), with Intriguing Effects on Neuropathic Pain
Ingår i In Neuropeptides in Neuroprotection and Neuroregeneration., s. 253-270, 2012.
-
Synthesis of functionalized furopyrazines as restricted dipeptidomimetics
Ingår i Tetrahedron, s. 3019-3029, 2012.
DOI för Synthesis of functionalized furopyrazines as restricted dipeptidomimetics
-
Transmetallation Versus β-Hydride Elimination: The Role of 1,4 Benzoquinone in Chelation-Controlled Arylation Reactions with Arylboronic Acids
Ingår i Chemistry - A European Journal, s. 4714-4722, 2012.
DOI för Transmetallation Versus β-Hydride Elimination: The Role of 1,4 Benzoquinone in Chelation-Controlled Arylation Reactions with Arylboronic Acids Ladda ner fulltext (pdf) av Transmetallation Versus β-Hydride Elimination: The Role of 1,4 Benzoquinone in Chelation-Controlled Arylation Reactions with Arylboronic Acids
-
Trisubstituted Imidazoles as Mycobacterium tuberculosis Glutamine Synthetase Inhibitors
Ingår i Journal of Medicinal Chemistry, s. 2894-2898, 2012.
DOI för Trisubstituted Imidazoles as Mycobacterium tuberculosis Glutamine Synthetase Inhibitors Ladda ner fulltext (pdf) av Trisubstituted Imidazoles as Mycobacterium tuberculosis Glutamine Synthetase Inhibitors
-
From the First Selective Non-Peptide AT(2) Receptor Agonist to Structurally Related Antagonists
Ingår i Journal of Medicinal Chemistry, s. 2265-2278, 2012.
-
Virtual Screening Data Fusion Using Both Structure- and Ligand-Based Methods
Ingår i Journal of Chemical Information and Modeling, s. 225-232, 2012.
DOI för Virtual Screening Data Fusion Using Both Structure- and Ligand-Based Methods
-
Angiotensin II, a neuropeptide at frontier between endocrinology and neuroscience: is there a link between the angiotensin II type 2 receptor andAlzheimer’s disease?
Ingår i Frontiers in Endocrinology, s. Article 17-, 2011.
-
The dipeptide Phe-Phe amide attenuates signs of hyperalgesia, allodynia and nociception in diabetic mice using a mechanism involving the sigma receptor system
Ingår i Molecular Pain, s. 85-, 2011.
DOI för The dipeptide Phe-Phe amide attenuates signs of hyperalgesia, allodynia and nociception in diabetic mice using a mechanism involving the sigma receptor system Ladda ner fulltext (pdf) av The dipeptide Phe-Phe amide attenuates signs of hyperalgesia, allodynia and nociception in diabetic mice using a mechanism involving the sigma receptor system
-
Substitution of the phosphonic acid and hydroxamic acid functionalities of the DXR inhibitor FR900098: An attempt to improve the activity against Mycobacterium tuberculosis
Ingår i Bioorganic & Medicinal Chemistry Letters, s. 5403-5407, 2011.
-
Synthesis of Functionalized Cinnamaldehyde Derivatives by an Oxidative Heck Reaction and Their Use as Starting Materials for Preparation of Mycobacterium tuberculosis 1-Deoxy-D-xylulose-5-phosphate Reductoisomerase Inhibitors
Ingår i Journal of Organic Chemistry, s. 8986-8998, 2011.
DOI för Synthesis of Functionalized Cinnamaldehyde Derivatives by an Oxidative Heck Reaction and Their Use as Starting Materials for Preparation of Mycobacterium tuberculosis 1-Deoxy-D-xylulose-5-phosphate Reductoisomerase Inhibitors Ladda ner fulltext (pdf) av Synthesis of Functionalized Cinnamaldehyde Derivatives by an Oxidative Heck Reaction and Their Use as Starting Materials for Preparation of Mycobacterium tuberculosis 1-Deoxy-D-xylulose-5-phosphate Reductoisomerase Inhibitors
-
P2-P1 ' macrocyclization of P2 phenylglycine based HCV NS3 protease inhibitors using ring-closing metathesis
Ingår i Bioorganic & Medicinal Chemistry, s. 4917-4927, 2011.
-
Design, Synthesis, and X-ray Crystallographic Studies of alpha-Aryl Substituted Fosmidomycin Analogues as Inhibitors of Mycobacterium tuberculosis 1-Deoxy-D-xylulose 5-Phosphate Reductoisomerase
Ingår i Journal of Medicinal Chemistry, s. 4964-4976, 2011.
DOI för Design, Synthesis, and X-ray Crystallographic Studies of alpha-Aryl Substituted Fosmidomycin Analogues as Inhibitors of Mycobacterium tuberculosis 1-Deoxy-D-xylulose 5-Phosphate Reductoisomerase Ladda ner fulltext (pdf) av Design, Synthesis, and X-ray Crystallographic Studies of alpha-Aryl Substituted Fosmidomycin Analogues as Inhibitors of Mycobacterium tuberculosis 1-Deoxy-D-xylulose 5-Phosphate Reductoisomerase
-
Non-peptide AT2-receptor agonists
Ingår i Current opinion in pharmacology (Print), s. 187-192, 2011.
-
Potent Macrocyclic Inhibitors of Insulin-Regulated Aminopeptidase (IRAP) by Olefin Ring-Closing Metathesis
Ingår i Journal of Medicinal Chemistry, s. 3779-3792, 2011.
-
Hepatitis C protease inhibitors based on 2(1H)-pyrazinones
Ingår i Abstracts of Papers of the American Chemical Society, s. 116-MEDI-, 2010.
-
Discovery of Dipeptides with High Affinity to the Specific Binding Site for Substance P1-7
Ingår i Journal of Medicinal Chemistry, s. 2383-2389, 2010.
DOI för Discovery of Dipeptides with High Affinity to the Specific Binding Site for Substance P1-7
-
Selective angiotensin II AT(2) receptor agonists with reduced CYP 450 inhibition
Ingår i Bioorganic & Medicinal Chemistry, s. 4570-4590, 2010.
DOI för Selective angiotensin II AT(2) receptor agonists with reduced CYP 450 inhibition
-
Improved P2 phenylglycine-based hepatitis C virus NS3 protease inhibitors with alkenylic prime-side substituents
Ingår i Bioorganic & Medicinal Chemistry, s. 5413-5424, 2010.
-
Disulfide cyclized tripeptide analogues of angiotensin IV as potent and selective inhibitors of insulin-regulated aminopeptidase (IRAP)
Ingår i Journal of Medicinal Chemistry, s. 8059-8071, 2010.
-
Discovery of Achiral Inhibitors of the Hepatitis C Virus NS3 Protease based on 2(1H)-pyrazinones
Ingår i Bioorganic & Medicinal Chemistry, s. 6512-6525, 2010.
-
Synthesis and evaluation of a 11C-labelled angiotensin II AT2 receptor ligand
Ingår i Journal of labelled compounds & radiopharmaceuticals, s. 616-624, 2010.
DOI för Synthesis and evaluation of a 11C-labelled angiotensin II AT2 receptor ligand
-
Hepatitis C virus NS3 protease inhibitors: large, flexible molecules of peptide origin show satisfactory permeability across Caco-2 cells
Ingår i European Journal of Pharmaceutical Sciences, s. 556-563, 2009.
-
A straightforward microwave method for rapid synthesis of N-1, C-6 functionalized 3,5-dichloro-2(1H)-pyrazinones
Ingår i Organic and biomolecular chemistry, s. 2809-2815, 2009.
-
Functionalized 3-amino-imidazo[1,2-a]pyridines: A novel class of drug-like Mycobacterium tuberculosis glutamine synthetase inhibitors
Ingår i Bioorganic & Medicinal Chemistry Letters, s. 4790-4793, 2009.
-
Structural basis for the inhibition of Mycobacterium tuberculosis glutamine synthetase by novel ATP-competitive inhibitors
Ingår i Journal of Molecular Biology, s. 504-513, 2009.
DOI för Structural basis for the inhibition of Mycobacterium tuberculosis glutamine synthetase by novel ATP-competitive inhibitors Ladda ner fulltext (pdf) av Structural basis for the inhibition of Mycobacterium tuberculosis glutamine synthetase by novel ATP-competitive inhibitors
-
New developments in the discovery of agents to treat hepatitis C
Ingår i Current Topics in Medicinal Chemistry, s. 533-562, 2008.
DOI för New developments in the discovery of agents to treat hepatitis C
-
Ligands to the (IRAP)/AT4 receptor encompassing a 4-hydroxydiphenylmethane scaffold replacing Tyr2
Ingår i Bioorganic & Medicinal Chemistry, s. 6924-6935, 2008.
-
Evaluation of the amino acid binding site of Mycobacterium tuberculosis glutamine synthetase for drug discovery
Ingår i Bioorganic & Medicinal Chemistry, s. 5501-5513, 2008.
DOI för Evaluation of the amino acid binding site of Mycobacterium tuberculosis glutamine synthetase for drug discovery Ladda ner fulltext (pdf) av Evaluation of the amino acid binding site of Mycobacterium tuberculosis glutamine synthetase for drug discovery
-
Is it possible to increase hit rates in structure-based virtual screening by pharmacophore filtering?: An investigation of the advantages and pitfalls of post-filtering
Ingår i Journal of Molecular Graphics and Modelling, s. 1237-1251, 2008.
-
Chemistry and folding of photomodulable peptides: stilbene and thioaurone-type candidates for conformational switches
Ingår i Organic and biomolecular chemistry, s. 4356-4373, 2008.
-
Identification of Plasmodium falciparum spermidine synthase active site binders through structure-based virtual screening
Ingår i Journal of Medicinal Chemistry, s. 2777-2786, 2008.
-
Selective angiotensin II AT2 receptor agonists: Benzamide structure–activity relationships
Ingår i Bioorganic & Medicinal Chemistry, s. 6841-6849, 2008.
DOI för Selective angiotensin II AT2 receptor agonists: Benzamide structure–activity relationships
-
Wallinder, Charlotta
Design, Synthesis and Biological Evaluation of Selective Nonpeptide AT2 Receptor Agonists and Antagonists
2008.
-
β-Amino acid substitutions and structure-based CoMFA modeling of hepatitis C virus NS3 protease inhibitors
Ingår i Bioorganic & Medicinal Chemistry, s. 5590-5605, 2008.
-
Modeling binding modes of angiotensin II and pseudopeptide analogues to the AT2 receptor
Ingår i Journal of Molecular Graphics and Modelling, s. 991-1003, 2008.
DOI för Modeling binding modes of angiotensin II and pseudopeptide analogues to the AT2 receptor
-
Hepatitis C Virus NS3 Protease Inhibitors Comprising a Novel Aromatic P1 Moiety
Ingår i Bioorganic & Medicinal Chemistry, s. 2955-2967, 2008.
DOI för Hepatitis C Virus NS3 Protease Inhibitors Comprising a Novel Aromatic P1 Moiety
-
Virtual screening and bioassay study of novel inhibitors for dengue virus mRNA cap (nucleoside-2'O)-methyltransferase
Ingår i Bioorganic & Medicinal Chemistry, s. 7795-7802, 2007.
-
Resistance profiling of hepatitis C virus protease inhibitors using full-length NS3
Ingår i Antiviral Therapy, s. 733-740, 2007.
-
Evaluation of a diverse set of potential P1 carboxylic acid bioisosteres in hepatitis C virus NS3 protease inhibitors
Ingår i Bioorganic & Medicinal Chemistry, s. 4057-4068, 2007.
-
Mechanistic studies of electrophilic protease inhibitors of full length hepatic C virus (HCV) NS3
Ingår i Journal of enzyme inhibition and medicinal chemistry (Print), s. 191-199, 2007.
-
Focused hierarchical design of peptide libraries - follow the lead
Ingår i Journal of Chemometrics, s. 486-495, 2007.
DOI för Focused hierarchical design of peptide libraries - follow the lead
-
Microwave-enhanced alpha-arylation of a protected glycine in water: evaluation of 3-phenylglycine derivatives as inhibitors of the tuberculosis enzyme, glutamine synthetase
Ingår i Combinatorial chemistry & high throughput screening, s. 783-789, 2007.
-
Quantitative structure-activity relationships of pine weevil antifeedants, a multivariate approach
Ingår i Journal of Agricultural and Food Chemistry, s. 9365-9372, 2007.
-
Selective angiotensin II AT(2) receptor agonists devoid of the imidazole ring system
Ingår i Bioorganic & Medicinal Chemistry, s. 7166-7183, 2007.
DOI för Selective angiotensin II AT(2) receptor agonists devoid of the imidazole ring system
-
Small potent ligands to the insulin-regulated aminopeptidase (IRAP)/AT(4) receptor
Ingår i Journal of Peptide Science, s. 434-444, 2007.
DOI för Small potent ligands to the insulin-regulated aminopeptidase (IRAP)/AT(4) receptor
-
Sköld, Christian
Computational Modeling of the AT2 Receptor and AT2 Receptor Ligands: Investigating Ligand Binding, Structure–Activity Relationships, and Receptor-Bound Models
2007.
-
Synthesis of a new class of druglike angiotensin II C-terminal mimics with affinity for the AT2 receptor
Ingår i Journal of Medicinal Chemistry, s. 1711-1715, 2007.
-
Development of CoMFA models of affinity and selectivity to angiotensin II type-1 and type-2 receptors
Ingår i Journal of Molecular Graphics and Modelling, s. 145-153, 2007.
-
Phenylglycine as a Novel P2 Scaffold in Hepatitis C Virus NS3 Protease Inhibitors
Ingår i Bioorganic & Medicinal Chemistry, s. 1448-1474, 2007.
DOI för Phenylglycine as a Novel P2 Scaffold in Hepatitis C Virus NS3 Protease Inhibitors
-
Design, synthesis, and incorporation of a beta-turn mimetic in angiotensin II forming novel pseudopeptides with affinity for AT(1) and AT(2) receptors
Ingår i Journal of Medicinal Chemistry, s. 6133-6137, 2006.
-
Fast and selective synthesis of novel cyclic sulfamide HIV-1 purchase inhibitors under controlled microwave heating
Ingår i Tetrahedron, s. 4671-4675, 2006.
-
Ligand bias of scoring functions in structure-based virtual screening.
Ingår i J Chem Inf Model, s. 1334-43, 2006.
-
Improved CoMFA modeling by optimization of settings.
Ingår i J Chem Inf Model, s. 355-64, 2006.
-
Presentation of a structurally diverse and commercially available drug data set for correlation and benchmarking studies.
Ingår i J Med Chem, s. 6660-71, 2006.
-
Selective angiotensin II AT(2) receptor agonists: Arylbenzylimidazole structure-activity relationships
Ingår i Journal of Medicinal Chemistry, s. 7160-7168, 2006.
-
Exploration of acyl sulfonamides as carboxylic acid replacements in protease inhibitors of the hepatitis C virus full-length NS3
Ingår i Bioorganic & Medicinal Chemistry, s. 544-559, 2006.
-
Short pseudopeptides containing turn scaffolds with high AT(2) receptor affinity
Ingår i Bioorganic & Medicinal Chemistry, s. 5963-5972, 2006.
DOI för Short pseudopeptides containing turn scaffolds with high AT(2) receptor affinity
-
A New Structural Theme in C2-Symmetric HIV-1 Protease Inhibitors: ortho-Substituted P1/P1’ Side Chains
Ingår i Bioorganic & Medicinal Chemistry, s. 5303-5315, 2006.
-
New selective AT2 receptor ligands encompassing a γ-turn mimetic replacing the amino acid residues 4-5 of angiotensin II act as agonists
Ingår i Journal of Medicinal Chemistry, s. 4009-4024, 2005.
-
A new tool in peptide engineering: a photoswitchable stilbene-type beta-hairpin mimetic.
Ingår i Chemistry, s. 403-12, 2005.
-
Synthesis, biological evaluation, and modeling studies of inhibitors aimed at the malarial proteases plasmepsins I and II.
Ingår i Bioorg Med Chem, s. 5371-90, 2005.
-
Cyclic sulfamide HIV-1 protease inhibitors, with sidechains spanning from P2/P2' to P1/P1'.
Ingår i Bioorg Med Chem, s. 755-64, 2005.
-
Design, Synthesis, and Biological Evaluation of the First Selective Nonpeptide AT2 Receptor Agonist
Ingår i Journal of Medicinal Chemistry, s. 5995-6008, 2004.
-
First Reported Nonpeptide AT1 Receptor Agonist (L-162,313) Acts as an AT2 Receptor Agonist in Vivo
Ingår i Journal of Medicinal Chemistry, s. 1536-1546, 2004.
-
Mycobacterium tuberculosis ribose-5-phosphate isomerase has a known fold, but a novel active site.
Ingår i J Mol Biol, s. 799-809, 2004.
-
AT2-selective angiotensin II analogues containing tyrosine-functionalized 5,5-bicyclic thiazabicycloalkane dipeptide mimetics.
Ingår i J Med Chem, s. 6009-19, 2004.
-
Conformer- and alignment-independent model for predicting structurally diverse competitive CYP2C9 inhibitors.
Ingår i J Med Chem, s. 907-14, 2004.
-
Structural analysis of CYP2C9 and CYP2C5 and an evaluation of commonly used molecular modeling techniques.
Ingår i Drug Metab Dispos, s. 1218-29, 2004.
-
Synthesis and AT2 receptor-binding properties of angiotensin II analogues
Ingår i Journal of Peptide Research, s. 194-201, 2004.
DOI för Synthesis and AT2 receptor-binding properties of angiotensin II analogues
-
A Selective AT2 Receptor Ligand with a γ-Turn-Like Mimetic replacing the Amino Acid Residues 4-5 of Angiotensin II
Ingår i Journal of Medicinal Chemistry, s. 859-870, 2004.
-
Structure-activity relationships for the selectivity of hepatitis C virus NS3 protease inhibitors
Ingår i Biochimica et Biophysica Acta, s. 51-59, 2004.
-
Acyl sulfonamides as potent protease inhibitors of the hepatitis C virus full-length NS3 (protease-helicase/NTPase): a comparative study of different C-terminals
Ingår i Bioorganic & Medicinal Chemistry, s. 2551-2568, 2003.
-
Antitumor activity of the novel melphalan containing tripeptide J3 (L-prolyl-melphalanyl-p-L-fluorophenylalanine ethyl ester): Comparison with its m-L-sarcolysin analogue P2
Ingår i Molecular Cancer Therapeutics, s. 1331-1339, 2003.
-
-
Vinyl sulfide cyclized analogues of angiotensin II with high affinity and full agonist activity at the AT(1) receptor
Ingår i Journal of Medicinal Chemistry, s. 1767-1777, 2002.
-
Tetrapeptides as potent protease inhibitors of Hepatitis C Virus full-length NS3 (protease-helicase/NTPase)
Ingår i Bioorganic & Medicinal Chemistry, s. 3915-22, 2002.
-
Effects of cholesterol and model transmembrane proteins on drugpartitioning into lipid bilayers as analysed by immobilized-liposomechromatography.
Ingår i J Pharm Pharmacol, s. 1477-, 2001.
-
Inhibition of hepatitis C virus NS3 protease activity by product-based peptides is dependent on helicase domain
Ingår i Bioorganic & Medicinal Chemistry Letters, s. 203-206, 2001.
-
Characterization of a set of HIV-1 protease inhibitors using binding kinetics data from a biosensor-based screen
Ingår i Journal of Biomolecular Screening, s. 353-359, 2000.
-
An Improved Procedure for N- to C-Directed (Inverse) Solid-Phase Peptide Synthesis
Ingår i Journal of combinatorial chemistry, s. 496-507, 2000.
DOI för An Improved Procedure for N- to C-Directed (Inverse) Solid-Phase Peptide Synthesis
-
Inhibitors of the C(2)-symmetric HIV-1 protease: nonsymmetric binding of asymmetric cyclic sulfamide with ketoxime groups in the P2/P2' side chains
Ingår i Journal of Medicinal Chemistry, s. 4054-4061, 1999.
-
Unexpected binding mode of a cyclic sulfamide HIV-1 protease inhibitor
Ingår i Journal of Medicinal Chemistry, s. 898-902, 1997.
DOI för Unexpected binding mode of a cyclic sulfamide HIV-1 protease inhibitor
-
Synthesis of C-2 symmetric potential inhibitors of HIV-1 protease from D-mannitol
Ingår i Journal of carbohydrate chemistry, s. 555-569, 1996.
DOI för Synthesis of C-2 symmetric potential inhibitors of HIV-1 protease from D-mannitol